| 1 | 4-(methoxycarbonyl)benzyl 1H-indole-4-carboxylate | 88.91 | 5.5 g |
| 2 | 4-(methoxycarbonyl)benzyl 1H-indazole-4-carboxylate | 85.34 | 4.7 g |
| 3 | 2-chloro-5-(4-fluorophenyl)thiazole-4-carbonitrile | 97.97 | 2 g |
| 4 | 2-(5-((3-((2H-tetrazol-5-yl)methoxy)azetidin-1-yl)sulfonyl)-2-ethoxyphenyl)-5-methyl-7-propyl-4a,7-dihydroimidazo[5,1-f][1,2,4]triazin-4(3H)-one | 99.28 | 2 g |
| 5 | 2-((1-((4-ethoxy-3-(5-methyl-4-oxo-7-propyl-3,4,4a,7-tetrahydroimidazo[5,1-f][1,2,4]triazin-2-yl)phenyl)sulfonyl)azetidin-3-yl)oxy)acetonitrile | 99.76 | 2 g |
| 6 | 2-(5-((3-((1H-1,2,3-triazol-4-yl)methoxy)azetidin-1-yl)sulfonyl)-2-ethoxyphenyl)-5-methyl-7-propyl-4a,7-dihydroimidazo[5,1-f][1,2,4]triazin-4(3H)-one | 98.86 | 4.5 g |
| 7 | 2-(5-((3-aminoazetidin-1-yl)sulfonyl)-2-ethoxyphenyl)-5-methyl-7-propyl-4a,7-dihydroimidazo[5,1-f][1,2,4]triazin-4(3H)-one | 98.98 | 1.5 g |
| 8 | methyl 4-(3-(4-(6-((4-cyano-2-fluorobenzyl)oxy)pyridin-2-yl)piperidin-1-yl)prop-1-yn-1-yl)-3-((2-methoxyethoxy)methyl)benzoate | 96.43 | 0.5 g |
| 9 | methyl 4-(3-(4-(6-((4-cyano-2-fluorobenzyl)oxy)pyridin-2-yl)piperidin-1-yl)prop-1-yn-1-yl)-3-((4-methoxybutoxy)methyl)benzoate | 96.73 | 0.46 g |
| 10 | 4-(3-(4-(6-((4-cyano-2-fluorobenzyl)oxy)pyridin-2-yl)piperidin-1-yl)prop-1-yn-1-yl)-3-((2-methoxyethoxy)methyl)benzoic acid | 97.16 | 0.03 g |
| 11 | methyl 4-(3-(4-(6-((4-cyano-2-fluorobenzyl)oxy)pyridin-2-yl)piperidin-1-yl)prop-1-yn-1-yl)-3-((3-methoxypropoxy)methyl)benzoate | 95.65 | 0.05 g |
| 12 | 4-((3-((4-ethoxy-3-(5-methyl-4-oxo-7-propyl-3,4-dihydroimidazo[5,1-f][1,2,4]triazin-2-yl)phenyl)sulfonamido)azetidin-1-yl)methyl)-3-fluoro-N-hydroxybenzamide | 95.97 | 0.2 g |
| 13 | methyl 6-(((1-((4-ethoxy-3-(5-methyl-4-oxo-7-propyl-3,4-dihydroimidazo[5,1-f][1,2,4]triazin-2-yl)phenyl)sulfonyl)azetidin-3-yl)amino)methyl)nicotinate | \ | 0.44 g |
| 14 | 4-(methoxycarbonyl)benzyl 1H-indole-6-carboxylate | 97.47 | 1.6 g |
| 15 | 4-(methoxycarbonyl)benzyl 1H-indazole-6-carboxylate | 95.72 | 1.7 g |
| 16 | 2-(5-((3-((2H-tetrazol-5-yl)methyl)-3-hydroxyazetidin-1-yl)sulfonyl)-2-ethoxyphenyl)-5-methyl-7-propylimidazo[5,1-f][1,2,4]triazin-4(3H)-one | 96.12 | 6 g |
| 17 | 2,2-dimethyl-4-nitrobutanoic acid | \ | 2.5 g |
| 18 | 4-(methoxycarbonyl)benzyl 1H-indole-5-carboxylate | 95.04 | 2.4 g |
| 19 | 4-(methoxycarbonyl)benzyl 1H-indazole-5-carboxylate | 70 | 3 g |
| 20 | 2-(5-chloro-2-ethoxyphenyl)-5-methyl-7-propylimidazo[5,1-f][1,2,4]triazin-4(3H)-one | 79.236 | 0.9 g |
| 21 | 2-(2-ethoxy-5-iodophenyl)-5-methyl-7-propylimidazo[5,1-f][1,2,4]triazin-4(3H)-one | 98.575 | 5.3 g |
| 22 | 2-chloro-8-cyclopentyl-6-iodo-5-methylpyrido[2,3-d]pyrimidin-7(8H)-one | 94.943 | 2.2 g |
| 23 | N-(5-(4-aminobutyl)pyridin-2-yl)-5-fluoro-4-(4-methylpiperazin-1-yl)pyrimidin-2-amine | 99.207 | 1.1 g |
| 24 | 2-chloro-5-fluoro-4-(4-methylpiperazin-1-yl)pyrimidine | 93.522 | 6.1 g |
| 25 | 4-chloro-5-fluoro-N-(5-nitropyridin-2-yl)pyrimidin-2-amine | 87.86 | 3.4 g |
| 26 | 4-(3-(5-((4-(3-(dimethylamino)azetidin-1-yl)-5-fluoropyrimidin-2-yl)amino)pyridin-2-yl)-4,4-dimethyl-5-oxo-2-thioxoimidazolidin-1-yl)-2-(trifluoromethyl)benzonitrile | 100 | 0.12 g |
| 27 | 4-(3-((5-((5-fluoro-4-(4-methylpiperazin-1-yl)pyrimidin-2-yl)amino)pyridin-2-yl)methyl)-4,4-dimethyl-5-oxo-2-thioxoimidazolidin-1-yl)-2-(trifluoromethyl)benzonitrile | 90.453 | 0.1 g |
| 28 | methyl 4-(((1-((4-ethoxy-3-(5-methyl-4-oxo-7-propyl-3,4-dihydroimidazo[5,1-f][1,2,4]triazin-2-yl)phenyl)sulfonyl)azetidin-3-yl)amino)methyl)-3-fluorobenzoate | 99.188 | 16 g |
| 29 | 2-(5-bromo-2-ethoxyphenyl)-5-methyl-7-propylimidazo[5,1-f][1,2,4]triazin-4(3H)-one | 97.927 | 1.9 g |
| 30 | 2-(5-amino-2-ethoxyphenyl)-5-methyl-7-propylimidazo[5,1-f][1,2,4]triazin-4(3H)-one | 85.65 | 33.4 g |
| 31 | methyl 1-(5-bromopyridin-2-yl)piperidine-4-carboxylate | 100 | 16.2 g |
| 32 | 3-(2-((3-(4-(ethoxycarbonyl)phenoxy)phenyl)amino)-2-oxoethyl)-1H-indole-2-carboxylic acid | 90 | 310 mg |
| 33 | methyl 3'-nitro-[1,1'-biphenyl]-3-carboxylate | 92 | 630 mg |
| 34 | 3-(2-((3'-(1-methoxyvinyl)-[1,1'-biphenyl]-3-yl)amino)-2-oxoethyl)-1H-indole-2-carboxylic acid | 93 | 270 mg |
| 35 | 3-(2-((3-(2-(methoxycarbonyl)phenoxy)phenyl)amino)-2-oxoethyl)-1H-indole-2-carboxylic acid | 92 | 150 mg |
| 36 | methyl 4,6-dichloropicolinate | 100 | 120 mg |
| 37 | (R)-4-(5-chloropyrazolo[1,5-a]pyrimidin-7-yl)-3-methylmorpholine | 100 | 120 mg |
| 38 | (S)-4-(3,6-dichloropyridazin-4-yl)-3-methylmorpholine | 94 | 110 mg |
| 39 | 3-(6-chloro-5-morpholinopyridazin-3-yl)-8-oxa-3-azabicyclo[3.2.1]octane | 99 | 120 mg |
| 40 | 5-chloro-7-(cyclopropylsulfonyl)pyrazolo[1,5-a]pyrimidine | 98 | 110 mg |
| 41 | 5-bromopyrazolo[1,5-a]pyridine | 100 | 120 mg |
| 42 | (R)-4-(7-iodopyrazolo[1,5-a]pyrimidin-5-yl)-3-methylmorpholine | 90 | 108 mg |
| 43 | 4-bromo-3,6-dichloropyridazine | 90 | 104 mg |
| 44 | (1R,5S)-3-(4-((R)-3-methylmorpholino)-7-(1H-pyrazol-3-yl)imidazo[1,5-b]pyridazin-2-yl)-8-oxa-3-azabicyclo[3.2.1]octane | 85 | 111 mg |
| 45 | (1R,5S)-3-(pyrazolo[1,5-a]pyrimidin-5-yl)-8-oxa-3-azabicyclo[3.2.1]octane | 95 | 108 mg |
| 46 | 4-(3,6-dichloropyridazin-4-yl)-2-methylmorpholine | 90 | 106 mg |
| 47 | N-((6-(8-oxa-3-azabicyclo[3.2.1]octan-3-yl)-4-(2-methylmorpholino)pyridazin-3-yl)methyl)-1H-pyrazole-5-carboxamide | 90 | 133 mg |
| 48 | 8-chloro-2-morpholino-1,7-naphthyridin-4-ol | 90 | 101 mg |
| 49 | 3,6-dichloro-4-(piperidin-1-yl)pyridazine | 95 | 105 mg |
| 50 | 7-benzyl-3-chloroisoquinoline | 95 | 102 mg |
| 51 | 2-(2,6-dioxopiperidin-3-yl)-5-(4-(hydroxymethyl)piperidin-1-yl)isoindoline-1,3-dione | 90 | 109 mg |
| 52 | 3-(6-chloro-5-(3,3-dimethylmorpholino)pyridazin-3-yl)-8-oxa-3-azabicyclo[3.2.1]octane | 90 | 133 mg |
| 53 | 2-(2,6-dioxopiperidin-3-yl)-5-(3-(hydroxymethyl)azetidin-1-yl)isoindoline-1,3-dione | 90 | 112 mg |
| 54 | 5-(3,6-dihydro-2H-pyran-4-yl)pyrazolo[1,5-a]pyrimidine | 90 | 120 mg |
| 55 | N-(2,3-dihydro-1H-inden-4-yl)pivalamide | 90 | 145 mg |
| 56 | N-(5-bromo-2,3-dihydro-1H-inden-4-yl)pivalamide | 90 | 130 mg |
| 57 | 1-(2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindolin-5-yl)piperidine-4-carbaldehyde | 90 | 119 mg |
| 58 | piperidin-4-yl 4-methylbenzenesulfonate hydrochloride | 90 | 126 mg |
| 59 | 2-(2,6-dioxopiperidin-3-yl)-5-(4-((4-hydroxypiperidin-1-yl)methyl)piperidin-1-yl)isoindoline-1,3-dione | 90 | 103 mg |
| 60 | 2-(2,6-dioxopiperidin-3-yl)-5-fluoroisoindoline-1,3-dione | 90 | 136 mg |
| 61 | (R)-4-(5-chloropyrazolo[1,5-a]pyrimidin-7-yl)-3-methylmorpholine | 95 | 103 mg |
| 62 | methyl 3'-(methylsulfonyl)-[1,1'-biphenyl]-4-carboxylate | 92 | 516 mg |
| 63 | 1-(4-([1,1'-biphenyl]-4-yloxy)-2-bromophenyl)ethan-1-one | 90 | 140 mg |
| 64 | 3-(4-nitrophenoxy)aniline | 99 | 588 mg |
| 65 | methyl 3-methyl-1H-indole-2-carboxylate | 100 | 130 mg |
| 66 | methyl 6-(pyridin-4-yl)-1H-indole-2-carboxylate | 95 | 310 mg |
| 67 | methyl 6-(benzyloxy)-1H-indole-2-carboxylate | 91 | 120 mg |
| 68 | 4-(3-nitrophenoxy)-1,1'-biphenyl | 99 | 180 mg |
| 69 | methyl 7-bromo-4-fluoro-3-(2-methoxy-2-oxoethyl)-1H-indole-2-carboxylate | 100 | 140 mg |
| 70 | 3-(carboxymethyl)-6-phenethoxy-1H-indole-2-carboxylic acid | 97 | 128 mg |
| 71 | methyl 2-amino-[1,1'-biphenyl]-4-carboxylate | 96 | 235 mg |
| 72 | 4-iodo-3-(trifluoromethyl)-1H-pyrazole | 100 | 170 mg |
| 73 | (R)-4-(3,6-dichloropyridazin-4-yl)-3-methylmorpholine | 98.28 | 200 mg |
| 74 | 3,6-dichloro-N-((5-methylimidazo[1,2-a]pyridin-2-yl)methyl)pyridazin-4-amine | 100 | 114 mg |
| 75 | ethyl 5-((tert-butoxycarbonyl)amino)pyrazolo[1,5-a]pyridine-3-carboxylate | 98.84 | 150 mg |
| 76 | 3-(2,6-difluoro-4-iodopyridin-3-yl)-N-(1-(tetrahydro-2H-pyran-2-yl)-1H-pyrazol-3-yl)propanamide | 98.77 | 185 mg |
| 77 | 3-(6-chloro-5-(4,4-difluoropiperidin-1-yl)pyridazin-3-yl)-8-oxa-3-azabicyclo[3.2.1]octane | 96.34 | 135 mg |
| 78 | (2S,6R)-4-(3,6-dichloropyridazin-4-yl)-2,6-dimethylmorpholine | 99.53 | 670 mg |
| 79 | tert-butyl 4-(5-chloropyrazolo[1,5-a]pyrimidin-7-yl)-3,6-dihydropyridine-1(2H)-carboxylate | 99.09 | 820 mg |
| 80 | 3-(2,4-difluoro-6-iodophenyl)propanoic acid | 92.14 | 1000 mg |
| 81 | 8-bromo-2,4-dichloro-1,5-naphthyridine | 95.72 | 270 mg |
| 82 | methyl 2-amino-4-bromo-3,5-difluorobenzoate | 90 | 2.7 g |
| 83 | 4-(4-aminophenoxy)benzenesulfonamide | 90 | 755 mg |
| 84 | 4-((4-chlorophenoxy)methyl)aniline | 90 | 3.97 g |
| 85 | 3'-amino-[1,1'-biphenyl]-3-sulfonamide | 90 | 4.91 g |
| 86 | tert-butyl 4-(3-bromobenzoyl)piperazine-1-carboxylate | 90 | 2.43 g |
| 87 | methyl 6-(benzyloxy)-3-(2-methoxy-2-oxoethyl)-1H-indole-2-carboxylate | 90 | 135 mg |
| 88 | 3-chloro-7-vinylisoquinoline | 90 | 800 mg |
| 89 | 2-(2,6-dioxopiperidin-3-yl)-4-fluoroisoindoline-1,3-dione | 90 | 330 mg |
| 90 | 2-(2,6-dioxopiperidin-3-yl)-4-hydroxyisoindoline-1,3-dione | 90 | 520 mg |
| 91 | ([1,1'-biphenyl]-3-ylmethyl)triphenylphosphonium bromide | 98.5 | 1.543 g |
| 92 | (4-phenoxybenzyl)triphenylphosphonium bromide | 97.2 | 344 mg |
| 93 | 1-(tert-butyl) 2-methyl 3-formyl-1H-indole-1,2-dicarboxylate | 93.5 | 1.167 g |
| 94 | methyl 3-formyl-1H-indole-2-carboxylate | 93.2 | 102 mg |
| 95 | 2-(2,6-dioxopiperidin-3-yl)-5-methylisoindoline-1,3-dione | 86.4 | 242 mg |
| 96 | ((4'-(methoxycarbonyl)-[1,1'-biphenyl]-2-yl)methyl)triphenylphosphonium bromide | 94.3 | 1.215 g |
| 97 | methyl 6-formyl-1H-indole-2-carboxylate | 95.6 | 777 mg |
| 98 | methyl 3'-nitro-[1,1'-biphenyl]-2-carboxylate | 96.5 | 243 mg |
| 99 | methyl (E)-3-(4-(([1,1'-biphenyl]-3-yloxy)methyl)phenyl)-2-azidoacrylate | 83.6 | 221 mg |
| 100 | 4-(benzyloxy)-2-nitrobenzenediazonium tetrafluoroborate | 84.3 | 1.744 g |
| 101 | 6-(benzyloxy)-3-(carboxymethyl)-1H-indole-2-carboxylic acid | 98.7 | 230 mg |
| 102 | methyl 5-(pyridin-4-yl)-1H-indole-2-carboxylate | 100 | 215 mg |
| 103 | methyl 4-amino-5-bromo-1,2-dihydropyridazine-3-carboxylate | 99.157 | 230 mg |
| 104 | 2-(methoxycarbonyl)-1H-indole-6-carboxylic acid | 97.1 | 222 mg |
| 105 | 2,4-dichloro-7-methoxy-1,8-naphthyridine | 86.6 | 180 mg |
| 106 | 3-methylthiomorpholine 1,1-dioxide
hydrogen chloride | 98.2 | 200 mg |
| 107 | 3,3'-(3-iodopyrazolo[1,5-a]pyrimidine-5,7-diyl)bis(6-oxa-3-azabicyclo[3.1.1]heptane) | 98.3 | 100 mg |
| 108 | 4-([1,1'-biphenyl]-4-yloxy)benzaldehyde | 98 | 160 mg |
| 109 | 1-(tert-butyl) 2-methyl 6-bromo-1H-indole-1,2-dicarboxylate | 100 | 180 mg |
| 110 | methyl 6-bromo-1H-indole-2-carboxylate | 89 | 140 mg |
| 111 | methyl 6-([1,1'-biphenyl]-4-yloxy)-1H-indole-2-carboxylate | 99 | 100 mg |
| 112 | 4-([1,1'-biphenyl]-3-yloxy)benzaldehyde | 100 | 450 mg |
| 113 | 4-amino-3-nitrobenzaldehyde | 98 | 120 mg |
| 114 | 3-(carboxymethyl)-1H-indole-2-carboxylic acid | 100 | 130 mg |
| 115 | 3-(carboxymethyl)-1-isobutylindoline-2-carboxylic acid | 100 | 130 mg |
| 116 | 4-(3-nitrobenzyl)morpholine | 100 | 250 mg |
| 117 | 6-chloro-3-fluoro-5-vinylpyridin-2-amine | 95 | 110 mg |
| 118 | 3-(4-aminophenoxy)benzenesulfonamide | 90 | 11.2 g |
| 119 | 4-(difluoromethoxy)-3-isopropoxybenzoic acid | 86.78 | 1.981 g |
| 120 | 2-(3-methylisothiazol-5-yl)isoindoline-1,3-dione | 91.94 | 2.232 g |
| 121 | N-((1H-1,2,4-triazol-3-yl)methyl)-2-ethoxybenzamide
Molecular Weight: 246.27 | 87.14 | 1.025 g |
| 122 | 3-(benzyloxy)-4-(difluoromethoxy)benzamide | 88.43 | 456 mg |
| 123 | 4-(3-(2-(2,4-difluorophenyl)-1,1-difluoro-2-hydroxy-3-(2H-tetrazol-2-yl)propyl)bicyclo[1.1.1]pentan-1-yl)phenol | 83.68 | 419 mg |
| 124 | methyl 5-cyanoquinoline-6-carboxylate | 98.97 | 1.298 g |
| 125 | 6-aminoquinoline-5-carbonitrile | 98.09 | 2.017 g |
| 126 | 2-ethoxy-N-(prop-2-yn-1-yl)benzamide | 99.04 | 6.228 g |
| 127 | 7a,9,10,11,12,12a-hexahydro-8H-[1,4]diazepino[5',6':4,5]thieno[3,2-f]quinolin-8-one | 100 | 466 mg |
| 128 | (2-fluoro-6-methoxypyridin-3-yl)boronic acid | 94.8 | 1080 mg |
| 129 | 3-bromo-5-(naphthalen-1-yl)pyridine | 96.3 | 1010 mg |
| 130 | ethyl 2-(7-methoxy-2-(trifluoromethyl)pyrazolo[1,5-a]pyridin-4-yl)oxazole-5-carboxylate | 97.3 | 165 mg |
| 131 | 4-bromo-2-ethoxyphenol | 92.71 | 3470 mg |
| 132 | 2-(7-methoxy-3H-spiro[benzofuran-2,1'-cyclopentan]-4-yl)-4,4,5,5-tetramethyl-1,3,2-dioxaborolane | 97.28 | 12.182 g |
| 133 | 2-(8-methoxy-2,2-dimethylchroman-5-yl)-4,4,5,5-tetramethyl-1,3,2-dioxaborolane | 87.42 | 1.372 g |
| 134 | 5-bromo-2-methoxyphenol | 100 | 2.171 g |
| 135 | 5-iodo-7-methoxy-3-methyl-3H-imidazo[4,5-b]pyridine | 96 | 168 mg |
| 136 | 2-bromo-6-fluoro-4-(trifluoromethyl)benzoic acid | 100 | 1.9 g |
| 137 | tert-butyl (4-bromo-2,2,5-trifluoro-1-oxido-3-oxo-2,3-dihydro-1l4-benzo[b]thiophen-1-ylidene)carbamate | 100 | 2.2 g |
| 138 | 5-bromo-8-methoxy-2-(trifluoromethyl)quinoline | 96.32 | 25.961 g |
| 139 | 5-(2-methoxyphenyl)-1,3,4-oxadiazol-2-amine | 95 | 4.3 g |
| 140 | 2-(5-amino-3-methyl-1H-pyrazol-1-yl)-6-propylpyrimidin-4(3H)-one | 95 | 1.2 g |
| 141 | 6-chloro-N-cyclohexyl-2-(pyridin-2-yl)pyrimidin-4-amine | 95 | 4.1 g |
| 142 | N-(5-bromoquinolin-8-yl)-4-methylbenzenesulfonamide | 90 | 640 mg |
| 143 | 3-chloro-6-(methylthio)-N-(tetrahydro-2H-pyran-4-yl)pyrazine-2-carboxamide | 95 | 360 mg |
| 144 | 3-chloro-N-(5-(2-methoxyphenyl)-1,3,4-oxadiazol-2-yl)-N-methylbenzamide | 95 | 70 mg |
| 145 | N-(3-methyl-1-(6-oxo-4-propyl-1,6-dihydropyrimidin-2-yl)-1H-pyrazol-5-yl)thiazole-2-carboxamide | 95 | 188 mg |
| 146 | 5-(2-methoxyphenyl)-N-(1-methyl-1H-benzo[d]imidazol-2-yl)-1,3,4-oxadiazol-2-amine | 93 | 132 mg |
| 147 | N-(5-(2-methoxyphenyl)-1,3,4-oxadiazol-2-yl)tetrahydro-2H-pyran-4-carboxamide | 95 | 50 mg |
| 148 | N-(5-(2-methoxyphenyl)-1,3,4-oxadiazol-2-yl)isobutyramide | 94 | 134 mg |
| 149 | N-(5-bromoquinolin-8-yl)tetrahydro-2H-pyran-4-sulfonamide | 95 | 72 mg |
| 150 | 2-(pyridin-2-yl)pyrimidine-4,6-diol | 90 | 4.1 g |
| 151 | 5-bromo-6-nitroquinoline | 90 | 1.3 g |
| 152 | 6,7-dimethoxy-2-methylquinazolin-4-ol | 100 | 11.3 g |
| 153 | 7-(benzyloxy)-6-methoxy-2-methylquinazolin-4-ol | 75 | 3.2 g |
| 154 | tert-butyl (S)-3-((7-methoxy-2-methyl-4-(((R)-1-(3-nitro-5-(trifluoromethyl)phenyl)ethyl)amino)quinazolin-6-yl)oxy)pyrrolidine-1-carboxylate | 97 | 4.6 g |
| 155 | (S)-tetrahydrofuran-3-yl methanesulfonate | \ | 3.5 g |
| 156 | tert-butyl (R)-3-((methylsulfonyl)oxy)pyrrolidine-1-carboxylate | \ | 28.3 g |
| 157 | 4-(benzyloxy)-5-hydroxy-2-nitrobenzoic acid | 85 | 9.5 g |
| 158 | 2-(3-azido-2-hydroxypropyl)isoindoline-1,3-dione | 100 | 1.2 g |
| 159 | 2-hydroxy-N-(4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)acetamide | 94 | 136 mg |
| 160 | 4-(bis(4-methoxybenzyl)amino)-1,3-dihydro-2H-imidazo[4,5-c]quinolin-2-one | 99 | 110 mg |
| 161 | 4-amino-1-(3-fluoro-4-(pyrrolidin-1-ylmethyl)benzyl)-1,3-dihydro-2H-imidazo[4,5-c]quinolin-2-one | 98 | 105 mg |
| 162 | 4-(2-(dimethylamino)ethoxy)benzonitrile | 93 | 171 mg |
| 163 | 2-(ethylthio)-1-(4-(pyrrolidin-1-ylmethyl)benzyl)-1H-imidazo[4,5-c]quinolin-4-amine | 97 | 75 mg |
| 164 | tert-butyl 4-((5-cyanothiophen-2-yl)methyl)piperazine-1-carboxylate | 99 | 105 mg |
| 165 | 6-butoxy-1-(4-(pyrrolidin-1-ylmethyl)benzyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine | 100 | 110 mg |
| 166 | ethyl (Z)-4-((phenyldiazenyl)methyl)benzoate | 93 | 135 mg |
| 167 | 2-(chloromethyl)isoindoline-1,3-dione | 90 | 4.5 g |
| 168 | 2-(chloromethyl)isoindoline-1,3-dione | 90 | 8.0 g |
| 169 | 2-(chloromethyl)isoindoline-1,3-dione | 90 | 6.9 g |
| 170 | 2,2'-(pyridin-2-ylmethylene)diphenol | 98 | 7.4 g |
| 171 | 2,2'-(pyridin-2-ylmethylene)diphenol | 98 | 1.5 g |
| 172 | benzyl(2-bromoethyl)sulfane | 90 | 5.7 g |
| 173 | 2-(chloromethyl)-1H-benzo[d]imidazole | 90 | 4.28 g |
| 174 | 5-fluoro-3-nitropicolinonitrile | 95 | 9.7 g |
| 175 | 5-bromo-3-(1,3-dioxolan-2-yl)-2-fluoropyridine | 94 | 2.28 g |
| 176 | 4-fluoroquinoline | 94 | 2.9 g |
| 177 | 2-cyclobutylacetonitrile | \ | 8.24 g |
| 178 | methyl (E)-4-bromo-3-((2-methyl-3-phenylallyl)oxy)benzoate | \ | 4.295 g |
| 179 | (Z)-N-((methylsulfonyl)oxy)acetimidoyl chloride | \ | 8.44 g |
| 180 | 3-benzyl-3-methyl-2,3-dihydrobenzofuran-6-carboxylic acid | 96 | 556 mg |
| 181 | 2-((5-bromo-2-nitrophenyl)amino)-N-(2-hydroxyethyl)acetamide | 95 | 110 mg |
| 182 | tert-butyl 4-(cyanomethylene)piperidine-1-carboxylate | 95 | 100 mg |
| 183 | potassium (3,5-dimethylisoxazol-4-yl)trifluoroborate | 95 | 19 g |
| 184 | methyl 2-(2,6-dioxopiperidin-3-yl)-1-oxoisoindoline-5-carboxylate | 90 | 219.84 mg |
| 185 | ethyl (E)-3-(3,5-dichlorophenyl)acrylate | 90 | 1986.44 mg |
| 186 | 3-(1-oxo-5-vinylisoindolin-2-yl)piperidine-2,6-dione | 90 | 831.19 mg |
| 187 | 3-(4-methoxybenzyl)imidazolidine-2,4-dione | 90 | 4484.23 mg |
| 188 | 5-(4-chlorophenyl)-1,3,4-oxadiazol-2-amine | 90 | 39.13 mg |
| 189 | 2-oxo-2-(pyridin-3-yl)acetic acid | 90 | 1428.28 mg |
| 190 | 2,2,5-tribromo-2,3-dihydro-1H-inden-1-one | 90 | 1622.07 mg |
| 191 | 2,5-dibromo-2,3-dihydro-1H-inden-1-one | 90 | 3929.72 mg |
| 192 | 3-bromopiperidine-2,6-dione | 90 | 321.23 mg |
| 193 | (E)-2-styrylthiophene | 90 | 3319.16 mg |
| 194 | 1-oxo-2,3-dihydro-1H-indene-5-carbonitrile | 90 | 1328.26 mg |
| 195 | 2-chloro-1-(3-hydroxyazetidin-1-yl)ethan-1-one | 95 | 2.73 g |
| 196 | 2-((2-cyclopropyl-8-fluoro-6-(4-(2-oxopropyl)piperazin-1-yl)quinolin-4-yl)(ethyl)amino)-4-(4-fluorophenyl)thiazole-5-carbonitrile | 95 | 140 mg |
| 197 | 2-((2-cyclopropyl-8-fluoro-6-(4-(2-hydroxypropyl)piperazin-1-yl)quinolin-4-yl)(ethyl)amino)-4-(4-fluorophenyl)thiazole-5-carbonitrile | 97 | 75 mg |
| 198 | 6-bromo-2-cyclopropyl-8-fluoro-N-methylquinolin-4-amine | 97 | 566 mg |
| 199 | (9H-fluoren-9-yl)methyl (4-(chloromethyl)-2-methoxybenzyl)carbamate | 93 | 410 mg |
| 200 | tert-butyl (R)-(3-(benzyloxy)-2-hydroxypropyl)(2,4-dimethoxybenzyl)carbamate | 95 | 150 mg |
| 201 | tert-butyl (R)-(3-(benzyloxy)-2-hydroxypropyl)(2,4-dimethoxybenzyl)carbamate | 95 | 4.28 g |
| 202 | N-((4-bromophenyl)sulfonyl)-3-methylbutanamide | 95 | 12.0 g |
| 203 | methyl 5-(chloromethyl)-4'-(N-(3-methylbutanoyl)sulfamoyl)-[1,1'-biphenyl]-3-carboxylate | 99 | 1.35 g |
| 204 | methyl 2-((((9H-fluoren-9-yl)methoxy)carbonyl)amino)-4-oxo-4,5-dihydrothiophene-3-carboxylate | 98 | 370 mg |
| 205 | methyl 4-(benzyloxy)-2,2-dimethylbutanoate | 91 | 8.65 g |
| 206 | N-(3-(((2-chloro-5-iodopyrimidin-4-yl)amino)methyl)pyrazin-2-yl)-N-methylmethanesulfonamide | 72 | 1.44 g |
| 207 | benzyl 3,3-difluorocyclobutane-1-carboxylate | 80 | 17.4 g |
| 208 | 1-chloro-7-methoxyisoquinoline-6-carbonitrile | 95 | 1.36 g |
| 209 | methyl 3-bromo-5-(hydroxymethyl)benzoate | 98 | 51.45 g |
| 210 | 2-methoxybenzyl carbamimidothioate hydrochloride | 95 | 22.13 g |
| 211 | tert-butyl 7-(methyl(7-tosyl-7H-pyrrolo[2,3-d]pyrimidin-4-yl)amino)-2-azaspiro[3.5]nonane-2-carboxylate | 93 | 1000 mg |
| 212 | methyl 2-bromo-5H-pyrrolo[2,3-b]pyrazine-7-carboxylate | 100 | 210 mg |
| 213 | 2-methoxy-3-(1-methyl-1H-1,2,4-triazol-3-yl)aniline | 97 | 900 mg |
| 214 | 2-methoxy-3-(1-methyl-1H-1,2,4-triazol-5-yl)aniline | 95.7 | 500 mg |
| 215 | N-(3-methoxy-1,2,4-thiadiazol-5-yl)-6-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)-1,6-diazaspiro[3.5]nonane-1-carboxamide | 99 | 700 mg |
| 216 | 6-bromo-2-(2,6-dimethylpyridin-4-yl)-3-methyl-1H-indole | 95 | 8.14 g |
| 217 | 6-(3-isopropyl-5-(piperidin-4-yl)-1H-indol-2-yl)-7,8-dimethyl-[1,2,4]triazolo[1,5-a]pyridine hydrochloride | 95 | 1.05 g |
| 218 | 2-(4-(2-(7,8-dimethyl-[1,2,4]triazolo[1,5-a]pyridin-6-yl)-3-isopropyl-1H-indol-5-yl)piperidin-1-yl)acetamide | 93 | 1.27 g |
| 219 | 6-bromo-3-(piperidin-1-ylmethyl)-1H-pyrrolo[2,3-b]pyridine | 96 | 648 mg |
| 220 | tert-butyl (2-((4-(1-(1-oxo-1,2-dihydroisoquinolin-5-yl)-5-(trifluoromethyl)-1H-pyrazole-4-carboxamido)-6-(trifluoromethyl)pyridin-2-yl)oxy)ethyl)carbamate | 95 | 295 mg |
| 221 | tert-butyl (1R,5S)-3-(7-bromo-6-chloro-8-fluoroquinazolin-4-yl)-3,8-diazabicyclo[3.2.1]octane-8-carboxylate | 99 | 780 mg |
| 222 | methyl 2-(1,4-dioxaspiro[4.5]decan-8-yl)-5-(6-(trifluoromethyl)picolinamido)-2H-indazole-6-carboxylate | 95 | 35 mg |
| 223 | N-(6-(2-hydroxypropan-2-yl)-2-(4-oxocyclohexyl)-2H-indazol-5-yl)-6-(trifluoromethyl)picolinamide | 90 | 550 mg |
| 224 | tert-butyl 4-hydroxy-2-(methylthio)-5,8-dihydropyrido[3,4-d]pyrimidine-7(6H)-carboxylate | \ | 6.85 g+8.05 g |
| 225 | tert-butyl (5-bromo-2-chloro-4-methylpyridin-3-yl)(tert-butoxycarbonyl)carbamate | \ | 8.23 g+5.10 g |
| 226 | 2-((4-chloropyrimidin-5-yl)oxy)-5-fluoro-N,N-diisopropylbenzamide | \ | 9.62 g |
| 227 | tert-butyl (S)-10-bromo-11-chloro-8-(2-isopropylphenyl)-7-oxo-3,4,7,8,13,13a-hexahydropyrazino[2',1':3,4][1,4]oxazepino[5,6,7-de]quinazoline-2(1H)-carboxylate | \ | 1.47 g |
| 228 | tert-butyl (5-bromo-4-chloropyridin-3-yl)(tert-butoxycarbonyl)carbamate | \ | 5.93 g |
| 229 | 7-fluoro-8-methylnaphthalen-1-yl trifluoromethanesulfonate | \ | 13.79 g |
| 230 | methyl 2-((4-chloropyrimidin-5-yl)oxy)-5-fluorobenzoate | \ | 2.87 g |
| 231 | 7-bromo-5-fluoro-1-(2-isopropylphenyl)quinazoline-2,4(1H,3H)-dione | \ | 1.1 g |
| 232 | 6-amino-4-bromo-3-chloro-2-fluorobenzonitrile | \ | 2.55 g |
| 233 | 6-amino-4-bromo-3-chloro-2-fluorobenzonitrile | \ | 2.72 g |
| 234 | 2-amino-4-bromo-6-fluorobenzonitrile | \ | 6.2 g |
| 235 | 2-amino-4-bromo-6-fluorobenzonitrile | \ | 3 g |
| 236 | (R)-(1-((3-methylpyrrolidin-1-yl)methyl)cyclopropyl)methanol | \ | 0.72 g |
| 237 | (1-(morpholinomethyl)cyclopropyl)methanol | \ | 0.88 g |
| 238 | (1-(pyrrolidin-1-ylmethyl)cyclopropyl)methanol | \ | 9.83 g |
| 239 | (E)-1-(4-chloro-1-(1-(tetrahydro-2H-pyran-2-yl)-1H-indazol-5-yl)-1H-benzo[d][1,2,3]triazol-6-yl)-3-(dimethylamino)prop-2-en-1-one | \ | 0.26 g |
| 240 | tert-butyl (tert-butoxycarbonyl)(4-methyl-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyridin-3-yl)carbamate | \ | 1 g |
| 241 | 7-fluoro-8-methylnaphthalen-1-yl trifluoromethanesulfonate | \ | 1.7 g |
| 242 | methyl 2-((2S,6S)-6-methyl-4-((4-nitrophenyl)sulfonyl)piperazin-2-yl)acetate | \ | 17 g |
| 243 | 1-benzyl 4-(tert-butyl) (S)-2-(cyanomethyl)piperazine-1,4-dicarboxylate | \ | 3.8 g |
| 244 | methyl 2-((2S,6S)-6-methyl-4-((4-nitrophenyl)sulfonyl)piperazin-2-yl)acetate | \ | 5.2 g |
| 245 | (S)-1-((benzyloxy)carbonyl)-4-(tert-butoxycarbonyl)piperazine-2-carboxylic acid | \ | 180 mg |
| 246 | benzyl (S)-2-(cyanomethyl)piperazine-1-carboxylate | \ | 3.7 g |
| 247 | 2-amino-4-bromo-6-fluorobenzonitrile | \ | 6.2 g |
| 248 | 4-bromo-2,6-difluorobenzamide | \ | 5 g |
| 249 | 2-amino-3-methyl-5-propylpyrazolo[1,5-a]pyrimidin-7(4H)-one | \ | 6.8 g |
| 250 | 1-bromo-8-chloronaphthalene | \ | 5.18 g |
| 251 | 8-benzyl-1,3,8-triazaspiro[4.5]decane-2,4-dione | \ | 1.7 g |
| 252 | 4-bromo-2,6-difluoro-N-((2-isopropylphenyl)carbamoyl)benzamide | \ | 3.3 g |
| 253 | benzyl (2-chloro-9-isopropyl-9H-purin-6-yl)glycinate | \ | 0.86 g |
| 254 | tert-butyl 4-(3,3-dimethylpiperazin-1-yl)benzoate | \ | 37.7 g |
| 255 | 4-(3,3-dimethylpiperazin-1-yl)benzoic acid | \ | 10 g |
| 256 | 6-(2,6-dichloro-3,5-dimethoxyphenyl)-1H-pyrazolo[3,4-b]pyridin-3-amine | \ | 15 g |
| 257 | methyl 4-(benzyloxy)-5-methoxy-2-nitrobenzoate | \ | 10 g |
| 258 | tert-butyl 4-(4-((benzyloxy)carbonyl)piperazin-1-yl)-2-(methylsulfonyl)-5,8-dihydropyrido[3,4-d]pyrimidine-7(6H)-carboxylate | \ | 12 g |
| 259 | 2-(4-fluorobenzyl)-4,7-dihydro-5H-thieno[2,3-c]pyran-3-carboxylic acid | \ | 25 g |
| 260 | benzyl (4-bromo-2-cyanophenyl)carbamate | \ | 20 g |
| 261 | methyl 2-((2R,6R)-6-methyl-4-((4-nitrophenyl)sulfonyl)piperazin-2-yl)acetate | \ | 75 g |
| 262 | methyl 2-((2R,6R)-6-methyl-4-((4-nitrophenyl)sulfonyl)piperazin-2-yl)acetate | \ | 23 g |
| 263 | 4-bromo-2,6-difluorobenzamide | \ | 21.6 g |
| 264 | tert-butyl (2-bromo-9-isopropyl-9H-purin-6-yl)glycinate | \ | 50.5 g |
| 265 | 6-chloro-2-fluoro-9-isopropyl-9H-purine | \ | 31.6 g |
| 266 | tert-butyl (2-chloro-9-isopropyl-9H-purin-6-yl)glycinate | \ | 130 g |
| 267 | tert-butyl (2-bromo-9-isopropyl-9H-purin-6-yl)glycinate | \ | 164 g |
| 268 | methyl (E)-3-(2-([1,1'-biphenyl]-3-yl)vinyl)-6-bromo-1H-indole-2-carboxylate | 90 | 116 mg |
| 269 | 3-(carboxymethyl)benzofuran-2-carboxylic acid | 90 | 1.2 g |
| 270 | 2'-methyl-[1,1'-biphenyl]-3-amine | 90 | 150 mg |
| 271 | methyl 3-(2-methoxy-2-oxoethyl)benzofuran-2-carboxylate | 90 | 300 mg |
| 272 | 4-(o-tolyl)pyridin-2-amine | 90 | 150 mg |
| 273 | methyl (E)-6-bromo-3-(4-phenoxystyryl)-1H-indole-2-carboxylate | 90 | 108 mg |
| 274 | 3-vinyl-1,1'-biphenyl | 90 | 155 mg |
| 275 | 2-methyl-3'-vinyl-1,1'-biphenyl | 90 | 190 mg |
| 276 | 1-phenoxy-2-vinylbenzene | | 101 mg |
| 277 | 4-(([1,1'-biphenyl]-2-yloxy)methyl)-2-bromobenzoic acid | 95 | 120 mg |
| 278 | methyl 3-(2-hydroxyethyl)-1H-indole-2-carboxylate | 100 | 130 mg |
| 279 | methyl 2'-amino-[1,1'-biphenyl]-4-carboxylate | 95 | 130 mg |
| 280 | 3-(carboxymethyl)-1-ethyl-1H-indole-2-carboxylic acid | 100 | 100 mg |
| 281 | 2-nitro-5-phenoxypyridine | 99 | 130 mg |
| 282 | 1-(2-bromo-4-((2'-methyl-[1,1'-biphenyl]-3-yl)oxy)phenyl)ethan-1-one | 95 | 100 mg |
| 283 | methyl 6-benzyl-1H-indole-2-carboxylate | 96 | 100 mg |
| 284 | 2-(methoxycarbonyl)-1H-indole-6-carboxylic acid | 90 | 121 mg |
| 285 | 2-phenoxybenzaldehyde | 100 | 221mg |
| 286 | methyl 2-(2-([1,1'-biphenyl]-3-ylamino)-2-oxoethyl)-4-aminobenzoate | 90 | 125 mg |
| 287 | methyl 6-hydroxy-3-(2-methoxy-2-oxoethyl)-1H-indole-2-carboxylate | 90 | 140 mg |
| 288 | tert-butyl (6-(4-(hydroxymethyl)phenoxy)hexyl)carbamate | 90 | 164 mg |
| 289 | tert-butyl (4-(4-(hydroxymethyl)phenoxy)butyl)carbamate | 90 | 329 mg |
| 290 | 6-((4-((8-aminooctyl)oxy)benzyl)oxy)-3-(4-phenoxyphenethyl)-1H-indole-2-carboxylic acid | 90 | 45 mg |
| 291 | 6-((4-((8-aminooctyl)oxy)benzyl)oxy)-3-(2-oxo-2-((4-phenoxyphenyl)amino)ethyl)-1H-indole-2-carboxylic acid | 90 | 127 mg |
| 292 | 5-methyl-2-nitrobenzenediazonium | 90 | 500 mg |
| 293 | 4'-nitro-[1,1'-biphenyl]-4-ol | 94.5 | 593 mg |
| 294 | MC21-1687-033 | 90 | 111 mg |
| 295 | MC-4034-118 | 90 | 122 mg |
| 296 | MC211417-126 | 90 | 110 mg |
| 297 | MC21-1702-023 | 90 | 106mg |
| 298 | MC21-1702-027 | 90 | 110mg |
| 299 | MC21-1686-048 | 90 | 137mg |
| 300 | MC21-1686-033 | 90 | 106mg |
| 301 | MC21-1659-012 | 90 | 105mg |
| 302 | MC21-1659-040 | 90 | 103mg |
| 303 | ((benzyloxy)carbonyl)glycine | 100 | 3 g |
| 304 | 2-chloro-3-nitro-N-(4-(pyrrolidin-1-ylmethyl)benzyl)quinolin-4-amine | 92.7 | 1 g |
| 305 | 1-(4-aminobutyl)-2-(methylthio)-1H-imidazo[4,5-c]quinolin-4-amine | 99 | 200 mg |
| 306 | ethyl glycinate | 98 | 1.5 g |
| 307 | 2-(methylthio)-1-((5-(pyrrolidin-1-ylmethyl)quinolin-8-yl)methyl)-1H-imidazo[4,5-c]quinolin-4-amine | 98.3 | 89 mg |
| 308 | 5-methylquinoline-8-carbonitrile | 100 | 383 mg |
| 309 | 2-butoxy-6-chloro-N,N-bis(4-methoxybenzyl)-5-nitropyrimidin-4-amine | 100 | 337 mg |
| 310 | 8-bromo-5-methylquinoline | 96.2 | 314 mg |
| 311 | 2-(butylthio)-6-chloro-N4,N4-bis(4-methoxybenzyl)pyrimidine-4,5-diamine | 94.3 | 209 mg |
| 312 | (2-amino-4-(methoxycarbonyl)phenyl)boronic acid | 98.8 | 157 mg |
| 313 | N-(4-(4-amino-2-(methylthio)-1H-imidazo[4,5-c]quinolin-1-yl)butyl)-4-((2,5-dioxo-2,5-dihydro-1H-pyrrol-1-yl)methyl)cyclohexane-1-carboxamide | 91.6 | 55mg |
| 314 | methyl 4-carbamoyl-2-nitrobenzoate | 99 | 185 mg |
| 315 | tert-butyl 1-(9H-fluoren-9-yl)-3,7-dioxo-2,11,14-trioxa-4,8-diazaheptadecan-17-oate | 98.7 | 210mg |
| 316 | 3-nitroquinoline-2,4-diol | 99.6 | 250mg |
| 317 | (6-(4-methylpiperazin-1-yl)pyridin-3-yl)methanamine | 99.6 | 200mg |
| 318 | tert-butyl 4-(methoxy(methyl)carbamoyl)piperidine-1-carboxylate | 88 | 141 mg |
| 319 | methyl 4-(([1,1'-biphenyl]-3-yloxy)methyl)-2-bromobenzoate | 98 | 350 mg |
| 320 | 4-(([1,1'-biphenyl]-3-yloxy)methyl)-2-bromo-N-methoxy-N-methylbenzamide | 100 | 300 mg |
| 321 | 3-(carboxymethyl)-6-(trifluoromethyl)-1H-indole-2-carboxylic acid | 94 | 50 mg |
| 322 | 6-benzyl-3-(1-carboxyethyl)-1H-indole-2-carboxylic acid | 95 | 60 mg |
| 323 | 9H-benzo[4,5]imidazo[2,1-c][1,2,4]triazol-3-amine | 93 | 213mg |
| 324 | 1-(2,4-bis(methoxymethoxy)phenyl)ethan-1-one | 95 | 221 mg |
| 325 | (S)-2-((naphthalen-1-yloxy)methyl)oxirane | 97 | 221 mg |
| 326 | (R)-2-((naphthalen-1-yloxy)methyl)oxirane | 77 | 206 mg |
| 327 | 2-allyl-4-nitrophenol | 99 | 210 mg |
| 328 | pyrido[2,3-d]pyridazin-8(7H)-one | 85 | 202 mg |
| 329 | 2-chloro-1H-benzo[d]imidazole-1-carbonitrile | 99 | 221 mg |
| 330 | 3-(benzylamino)-1,1,1-trifluoropropan-2-ol | \ | 7.2 g |
| 331 | methyl N-(tert-butoxycarbonyl)-O-(tert-butyldiphenylsilyl)-D-serinate | \ | 8.9 g |
| 332 | methyl O-benzyl-N-(tert-butoxycarbonyl)-D-serinate | \ | 3.6 g |
| 333 | 2-chloro-5,6,7,8-tetrahydro-1,6-naphthyridine | \ | 6.5 g |
| 334 | (tert-butoxycarbonyl)-L-proline | \ | 8 g |
| 335 | tert-butyl piperidin-4-ylcarbamate | \ | 4.8 g |
| 336 | 4-(2-fluoropyridin-3-yl)-2-(methylthio)pyrimidine | 100 | 110 mg |
| 337 | 2-methoxy-5-methyl-4-(4-(4-methylpiperazin-1-yl)piperidin-1-yl)aniline | 100 | 200 mg |
| 338 | tert-butyl (S)-4-(2-hydroxyquinoxalin-6-yl)-2-methylpiperazine-1-carboxylate | 91 | 115 mg |
| 339 | 4-methylbenzyl carbamimidothioate | 93 | 120 mg |
| 340 | 5-bromo-7-methoxy-2-methyl-2H-indazole | 100 | 105 mg |
| 341 | 2,7-dimethylpyrazolo[1,5-a]pyridine-5-carbonitrile | 100 | 103 mg |
| 342 | (S)-6-(3-methylpiperazin-1-yl)benzo[d]thiazole | 98 | 110 mg |
| 343 | 5-bromo-7-methoxy-1-methyl-1H-indazole | 99 | 102 mg |
| 344 | 6-bromo-2-methylimidazo[1,2-a]pyrazine | 95 | 150 mg |
| 345 | tert-butyl (S)-4-(benzo[d]thiazol-6-yl)-2-methylpiperazine-1-carboxylate | 90 | 202 mg |
| 346 | 5-bromopyrazin-2-amine | 98 | 150 mg |
| 347 | tert-butyl (S)-4-(6-aminopyridazin-3-yl)-2-methylpiperazine-1-carboxylate | 99 | 100 mg |
| 348 | 7-methoxy-3-nitroquinolin-4-ol | 94 | 105mg |
| 349 | 2-bromo-6-chloro-4-methylpyridin-3-amine | 98 | 100 mg |
| 350 | ethyl 4-chloro-6-fluoro-7-methoxyquinoline-3-carboxylate | 98 | 110 mg |
| 351 | N-(4-bromo-2,6-difluorobenzyl)-7-methoxy-3-nitroquinolin-4-amine | 100 | 110 mg |
| 352 | 6-chloro-2,8-dimethylimidazo[1,2-b]pyridazine | 99 | 113 mg |
| 353 | tert-butyl (4-methoxypyridin-2-yl)carbamate | 97 | 100 mg |
| 354 | 5-bromo-7-methoxy-2-methyl-2H-pyrazolo[3,4-c]pyridine | 99 | 116 mg |
| 355 | 4-chloro-7-methoxy-3-nitroquinoline | 98 | 150 mg |
| 356 | N2-(4-chlorophenyl)-N6-cyclopropyl-3-nitropyridine-2,6-diamine | 100 | 3.0g |
| 357 | 3-(4-(benzyloxy)phenyl)-4-iodo-1H-pyrazole | 100 | 3.1g |
| 358 | ethyl 5-morpholinopyrazolo[1,5-a]pyrimidine-3-carboxylate | 91 | 2.9g |
| 359 | 6-chloro-2-iodo-N-(4-methoxybenzyl)pyrimidin-4-amine | 91.27 | 4.8g |
| 360 | 2-methoxy-4-methylbenzoic acid | 100 | 3.1g |
| 361 | benzyl 4-(tosyloxy)piperidine-1-carboxylate | 100 | 4.4g |
| 362 | 5-morpholinopyrazolo[1,5-a]pyrimidine-3-carboxylic acid | 100 | 0.9g |
| 363 | 3-aminopicolinonitrile | 100 | 1.3g |
| 364 | 5-bromo-2-methoxy-3-nitrobenzamide | 74.48 | 2.1g |
| 365 | ethyl 5-(2-oxa-5-azabicyclo[2.2.1]heptan-5-yl)pyrazolo[1,5-a]pyrimidine-3-carboxylate | 100 | 1.3g |
| 366 | 2-(5,6-dichloropyridin-3-yl)acetonitrile | 83.61 | 2.1g |
| 367 | 2-hydroxy-3-nitrobenzamide | 98.9 | 8.1g |
| 368 | 4-iodo-3-(4-phenoxyphenyl)-1H-pyrazole | 76.69 | 4.3g |
| 369 | 5-bromopicolinamide | 100 | 4.6g |
| 370 | 2-chloro-5-nitropyridin-4-amine | 100 | 4.5g |
| 371 | 3-aminopicolinamide | 97.42 | 4.9g |
| 372 | 5-nitroisothiazole-3-carboxylic acid | 100 | 5.2g |
| 373 | tert-butyl 3-(2,5-dioxo-4-(pyridin-2-yl)imidazolidin-4-yl)propanoate | 100 | 0.9g |
| 374 | 7-chloro-1,3,4,5-tetrahydro-2H-benzo[d]azepin-2-one | 100 | 2.6g |
| 375 | methyl 6-chloro-4-((3-((2,2,2-trifluoroacetamido)methyl)phenyl)thio)pyridazine-3-carboxylate | 100 | 0.3g |
| 376 | 3-aminopicolinamide | 100 | 1.0g |
| 377 | N-(5-bromo-8-(methylamino)-4a,8a-dihydropyrido[3,4-c]pyridazin-3-yl)cyclopropanecarboxamide | 100 | 0.2g |
| 378 | ethyl 5-amino-1-(4-methoxybenzyl)-1H-pyrazole-4-carboxylate | 100 | 0.8g |
| 379 | 4-bromo-2-ethoxy-6-nitroaniline | 100 | 2.9g |
| 380 | tert-butyl (5-(4-aminopyrimidin-2-yl)thiazol-2-yl)(pent-4-en-1-yl)carbamate | 100 | 2.0g |
| 381 | N4-(1-methylpiperidin-4-yl)-5-(trifluoromethyl)benzene-1,2,4-triamine | 94 | 0.9g |
| 382 | 5-bromo-2-hydroxy-4-methoxynicotinonitrile | 84 | 0.2g |
| 383 | 1H-indol-4-amine | 97.76 | 5.1g |
| 384 | tert-butyl (1-(pyrimidin-2-yl)butyl)carbamate | 100 | 3.0g |
| 385 | 1-(4-amino-5-nitropyridin-2-yl)piperidin-4-ol | 100 | 0.6g |
| 386 | tert-butyl (5-(4-aminopyridin-2-yl)thiazol-2-yl)(pent-4-en-1-yl)carbamate | 94 | 0.6g |
| 387 | 5-(hydroxymethyl)-2-methylphenol | 100 | 1.7g |
| 388 | 1-(2-chloro-5H-pyrrolo[2,3-d]pyrimidin-5-yl)propan-1-one | 100 | 0.9g |
| 389 | tert-butyl (5-(4-aminopyrimidin-2-yl)thiazol-2-yl)(pent-4-en-1-yl)carbamate | 100 | 2.1g |
| 390 | methyl 2-acrylamido-4-((tert-butoxycarbonyl)(2-(tosyloxy)propyl)amino)benzoate | 100 | 0.6g |
| 391 | N-(1-(4-bromobenzoyl)piperidin-4-yl)acetamide | 100 | 0.6g |
| 392 | 4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-5,6-dihydropyridin-2(1H)-one | 100 | 2.5g |
| 393 | 4-chloro-3-(6-(2-methyl-6-methylenemorpholino)-1H-imidazo[4,5-c]pyridin-2-yl)-3,4-dihydroquinolin-2(1H)-one | 40 | 1.2g |
| 394 | 2-methoxy-1-(pyrimidin-2-yl)ethan-1-amine | 100 | 1.3g |
| 395 | tert-butyl (2-methyl-1-(pyrimidin-2-yl)propyl)carbamate | 100 | 1.0g |
| 396 | cyclohexyl(pyrimidin-2-yl)methanamine | 85 | 3g |
| 397 | 2,6-difluoro-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenol | 85 | 1.2g |
| 398 | 8-(aminomethyl)-3-benzyl-2-hydroxy-4H-benzo[4,5]thiazolo[3,2-a]pyrimidin-4-one | 100 | 0.1g |
| 399 | N-(3-((6-(3-(2,6-dichloro-3,5-dimethoxyphenyl)ureido)pyrimidin-4-yl)amino)-1-methyl-2,3-dihydro-1H-pyrazol-4-yl)acrylamide | 100 | 0.5g |
| 400 | 2-Aminothiazole | 100 | 1.4g |
| 401 | 4-(4-cyclohexylpiperazin-1-yl)benzene-1,2-diamine | 75 | 1.1g |
| 402 | 4-(4-bromo-3-methoxyphenyl)-1-methyl-1H-pyrazole | 100 | 5.0g |
| 403 | 1-(3-bromopyridin-2-yl)piperidine-4-carbohydrazide | 100 | 1.4g |
| 404 | (4-bromophenyl)(3-(hydroxymethyl)cyclopentyl)methanone | 100 | 1.6g |
| 405 | 3-(3-bromo-2-methoxyphenyl)-1-methyl-1H-1,2,4-triazole | 100 | 5.5g |
| 406 | 7-bromo-3-methylene-3,4-dihydro-2H-pyrido[3,2-b][1,4]oxazine | 100 | 1.5g |
| 407 | (4-chloro-3-nitrophenyl)dimethylphosphine oxide | 100 | 4.3g |
| 408 | 4-bromo-9H-pyrido[3,4-b]indole | 84 | 4.4g |
| 409 | 2-((3-amino-4-nitrophenyl)amino)ethan-1-ol | 100 | 3.9g |
| 410 | tert-butyl (1-(3-methylpyridin-2-yl)ethyl)carbamate | 100 | 0.8g |
| 411 | 2-nitro-5-(2,2,6-trimethylmorpholino)aniline | 100 | 4.2g |
| 412 | 1-(4-amino-5-nitropyridin-2-yl)azetidin-3-ol | 100 | 0.8g |
| 413 | 5-(3-bromo-2-methoxyphenyl)-4,5-dihydrooxazole | 100 | 3.7g |
| 414 | 2-methoxy-5-nitropyridin-4-amine | 100 | 2.9g |
| 415 | 5-(4-chloro-2-fluoro-5-methoxyphenyl)-1-(difluoromethyl)-2-methyl-1,2-dihydro-3H-pyrazol-3-one | 100 | 2.7g |
| 416 | 2-methoxy-3-(1-methyl-1H-1,2,4-triazol-3-yl)phenol | 100 | 1.5g |
| 417 | N-(4-(1-methoxyvinyl)phenyl)acrylamide | 100 | 1.2g |
| 418 | 8-(trifluoromethyl)quinazolin-4-ol | 59 | 4.7g |
| 419 | ethyl 4-bromothiazole-5-carboxylate | 98 | 3.9g |
| 420 | 2-methoxy-4-morpholinobenzoic acid | 100 | 108g |
| 421 | 2-carbamoyl-1-(4-chloro-2-methylphenyl)-6-methoxy-1,2,3,4-tetrahydroisoquinolin-7-yl trifluoromethanesulfonate | 100 | 8.1g |
| 422 | 3-(trifluoromethyl)benzohydrazide | 100 | 8.9g |
| 423 | N-(4-bromobenzyl)-2,2,2-trifluoroacetamide | 100 | 10.9g |
| 424 | methyl 6-chloro-4-((2-(methylthio)phenyl)amino)nicotinate | 100 | 2.6g |
| 425 | 4-iodo-2-methoxynicotinaldehyde | 78 | 9.2g |
| 426 | 2-bromo-3,4-dichloro-5-methyl-6-nitroaniline | 100 | 7.3g |
| 427 | 4-fluoro-5-morpholinobenzene-1,2-diamine | 100 | 8g |
| 428 | 7-chloro-4-(4-methoxybenzyl)-2-methyl-5-oxo-4,5,6,7-tetrahydro-2H-pyrazolo[4,3-b]pyridine-6-carbaldehyde | 93.4 | 102.1g+37.5g |
| 429 | 5-bromo-2-methoxy-3-nitrobenzamide | 88.5 | 15.42g |
| 430 | 4-(benzyloxy)-2-naphthoic acid | 92.79 | 115.1g+52.4g |
| 431 | 4-bromophenol | 100 | 41.4g |
| 432 | 7-chloro-2-ethyl-4-(4-methoxybenzyl)-5-oxo-4,5-dihydro-2H-[1,2,3]triazolo[4,5-b]pyridine-6-carbaldehyde | 78 | 161.1g+88.9g |
| 433 | methyl 6-chloro-4-((2-(methylthio)phenyl)amino)nicotinate | 100 | 3.9g |
| 434 | tert-butyl 3-carbamoylazetidine-1-carboxylate | 100 | 7.6g |
| 435 | N-(3-bromobenzyl)-2,2,2-trifluoroacetamide | 100 | 7.5g |
| 436 | 5-bromothiazol-2-amine | 100 | 43.8g |
| 437 | 5-bromo-4-iodo-2-methoxynicotinaldehyde | 91 | 6.3g |
| 438 | 1-(2-chloro-7-(pent-4-en-2-yl)-7H-pyrrolo[2,3-d]pyrimidin-5-yl)propan-1-one | 100 | 15.1g |
| 439 | 4-Quinazolinamine, N-(3-chloro-4-fluorophenyl)-7-fluoro-6-nitro- | 99 | 4.4g |
| 440 | 7-nitro-1-tosyl-1H-indole | 95 | 8.5g |
| 441 | methyl 5-methyl-1H-pyrazole-3-carboxylate | 100 | 142.5g |
| 442 | 2-(4-hydroxy-3-nitrophenyl)acetic acid | 100 | 27.2g |
| 443 | 7-chloro-2-ethyl-4-(4-methoxybenzyl)-5-oxo-4,5-dihydro-2H-pyrazolo[4,3-b]pyridine-6-carbaldehyde | 100 | 3.4g |
| 444 | 6-chloro-4-methylpyridazin-3(2H)-one | 100 | 3.6g |
| 445 | N-(3-chloro-4-methoxy-2-nitrophenyl)acetamide | 100 | 3g |
| 446 | 2-fluoro-3-morpholino-6-nitroaniline | 80.7 | 10.7g |
| 447 | ethyl 5-morpholinopyrazolo[1,5-a]pyrimidine-3-carboxylate | 100 | 7.4g |
| 448 | 4-nitro-1H-indole | 93 | 45.3g |
| 449 | 5-(1-methoxyvinyl)-4-nitro-1H-pyrazole | 100 | 28g |
| 450 | tert-butyl (2-methyl-1-(pyridin-2-yl)propyl)carbamate | 100 | 16.9g |
| 451 | 5-([1,4'-bipiperidin]-1'-yl)-2-nitroaniline | 100 | 7.9g |
| 452 | tert-butyl (E)-3-(4-morpholinophenyl)acrylate | 99 | 1753mg |
| 453 | 2-(5-fluoro-1H-indol-3-yl)-2-oxoacetic acid | 99 | 982mg |
| 454 | 2-(7-chloro-1H-indol-3-yl)-2-oxoacetic acid | 99 | 484mg |
| 455 | 2-(7-fluoro-1H-indol-3-yl)-2-oxoacetic acid | 99 | 1006mg |
| 456 | 2-(5-methoxy-1H-indol-3-yl)-2-oxoacetic acid | 99 | 2001mg |
| 457 | tert-butyl (E)-3-(4-(4-methylpiperazin-1-yl)phenyl)acrylate | 99 | 2187mg |
| 458 | 2-(5-methyl-1H-indol-3-yl)-2-oxoacetic acid | 99 | 807mg |
| 459 | 2-(7-methyl-1H-indol-3-yl)-2-oxoacetic acid | 99 | 2089mg |
| 460 | 2-(6-methoxy-1H-indol-3-yl)-2-oxoacetic acid | 99 | 1877mg |
| 461 | 2-(6-methyl-1H-indol-3-yl)-2-oxoacetic acid | 99 | 924mg |
| 462 | 2-(5-chloro-1H-indol-3-yl)-2-oxoacetic acid | 99 | 297mg |
| 463 | 4-(piperidin-1-yl)benzaldehyde | 99 | 1657mg |
| 464 | 4-morpholinobenzaldehyde | 99 | 1786mg |
| 465 | 2-(4-methoxy-1H-indol-3-yl)-2-oxoacetic acid | 99 | 2231mg |
| 466 | 2-(4-chloro-1H-indol-3-yl)-2-oxoacetic acid | 99 | 1729mg |
| 467 | 5-phenyl-3,4-dihydronaphthalen-1(2H)-one | 99 | 103 mg |
| 468 | methyl 6-(benzyloxy)-1H-indole-2-carboxylate | 95 | 121 mg |
| 469 | methyl 3-(4-(cyclohexyloxy)phenethyl)-6-methoxy-1H-indole-2-carboxylate | 95 | 100 mg |
| 470 | 1-allyl-3-(cyclohexyloxy)benzene | 90 | 115 mg |
| 471 | methyl 6-phenoxy-1H-indole-2-carboxylate | 90 | 125 mg |
| 472 | methyl 6-(3-((tert-butyldimethylsilyl)oxy)propyl)-1H-indole-2-carboxylate | 95 | 130 mg |
| 473 | 3-vinyl-1,1'-biphenyl | 99 | 105 mg |
| 474 | 2-(2,6-difluoro-4-(methylthio)phenyl)-4,4,5,5-tetramethyl-1,3,2-dioxaborolane | 90 | 480 mg |
| 475 | (3,5-difluorophenyl)(methyl)sulfane | 90 | 220 mg |
| 476 | 3-(2-bromo-3-methylphenyl)propan-1-ol | 90 | 350 mg |
| 477 | 3'-bromo-2-methyl-1,1'-biphenyl | 90 | 587 mg |
| 478 | methyl 3-(2-hydroxyethyl)-6-methyl-1H-indole-2-carboxylate | 90 | 113 mg |
| 479 | 1-(benzyloxy)-4-(4-vinylphenoxy)benzene | 90 | 133 mg |
| 480 | 1-(4-vinylphenyl)piperidine | | 125 mg |
| 481 | phenyl(2-vinylphenyl)methanone | 95 | 265 mg |
| 482 | 3-(2-(2'-methyl-[1,1'-biphenyl]-3-yl)ethyl)-1H-indole-2-carboxylic acid | 98 | 50 mg |
| 483 | 3-(3-fluorophenyl)-1-vinylbenzene | 90 | 131 mg |
| 484 | 2-chloro-1-(3-vinylphenyl)benzene | 90 | 153 mg |
| 485 | 4-fluoro-1-(3-vinylphenyl)benzene | 90 | 204 mg |
| 486 | 4-(phenyloxy)-1-(prop-2-enyl)benzene | 90 | 134 mg |
| 487 | 4-{[3-(benzyloxy)phenyl]oxy}benzene-1-carbaldehyde | 90 | 143 mg |
| 488 | phenyl(4-vinylphenyl)methanone | 90 | 118mg |
| 489 | methyl 3-[(1E)-2-[3-(3-fluorophenyl)phenyl]vinyl]-1H-indole-2-carboxylate | 90 | 104mg |
| 490 | methyl 3-[(1E)-2-[3-(2-chlorophenyl)phenyl]vinyl]-1H-indole-2-carboxylate | 90 | 106mg |
| 491 | methyl 3-[(1E)-2-(4-{[3-(benzyloxy)phenyl]oxy}phenyl)vinyl]-1H-indole-2-carboxylate | 90 | 105mg |
| 492 | 3-[3-methyl-2-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]propan-1-ol | 90 | 105mg |
| 493 | 3-(4-bromo-3-methylphenyl)prop-2-yn-1-ol | 90 | 120mg |
| 494 | 3'-methoxy-2,3,4,5-tetrahydro-1,1'-biphenyl | 90 | 101 mg |
| 495 | 3-cyclohexylphenol | 98 | 156 mg |
| 496 | 4-((3-cyclohexylphenoxy)methyl)benzaldehyde | 90 | 182 mg |
| 497 | 3-cyclohexylaniline | 93 | 156mg |
| 498 | ethyl 2-(4-acetylphenyl)acetate | 98 | 186 mg |
| 499 | 4-(4-cyclohexylphenoxy)benzaldehyde | 96 | 203 mg |
| 500 | 4-(4-fluorophenoxy)benzaldehyde | 99 | 197 mg |
| 501 | methyl (E)-6-(3-((tert-butyldimethylsilyl)oxy)propyl)-3-(2-(2'-methyl-[1,1'-biphenyl]-3-yl)vinyl)-1H-indole-2-carboxylate | 95 | 169 mg |
| 502 | 2-bromo-5-phenyl-1,2,3,4-tetrahydronaphthalen-1-ol | 97 | 143 mg |
| 503 | methyl (E)-3-(3-bromostyryl)-1H-indole-2-carboxylate | 99 | 102 mg |
| 504 | methyl (E)-2-azido-3-(4-((3-cyclohexylphenoxy)methyl)phenyl)acrylate | 96 | 118 mg |
| 505 | 2-methyl-1-nitro-4-phenoxybenzene | 96 | 243 mg |
| 506 | methyl 3-(2-(2'-methyl-4-(3-((methylsulfonyl)oxy)propyl)-[1,1'-biphenyl]-3-yl)ethyl)-1H-indole-2-carboxylate | 90 | 56 mg |
| 507 | (R)-4-benzyl-3-((S)-2-(3-chloropropyl)pent-4-enoyl)oxazolidin-2-one | 90 | 135 mg |
| 508 | (S)-2-(3-chloropropyl)pent-4-en-1-ol | 90 | 110 mg |
| 509 | 5-allyl-1,3-dioxane | 90 | 120 mg |
| 510 | (S)-2-(tetrahydro-2H-pyran-3-yl)acetic acid | 90 | 65 mg |
| 511 | methyl 3-(2-(6-(3-hydroxypropyl)-2'-methyl-[1,1'-biphenyl]-3-yl)ethyl)-1H-indole-2-carboxylate | 95 | 100mg |
| 512 | methyl 6-bromo-3-(2-ethoxy-2-oxoethyl)-1H-indole-2-carboxylate | 100 | 110mg |
| 513 | 3'-ethynyl-4-fluoro-2-methyl-1,1'-biphenyl | 95 | 120mg |
| 514 | tert-butyl (4-(4-formylphenoxy)butyl)carbamate | 100 | 110mg |
| 515 | methyl 6-(3-(3-hydroxypropyl)phenoxy)-1H-indole-2-carboxylate | 98 | 140mg |
| 516 | 3-(3-hydroxypropyl)phenol | 95 | 120mg |
| 517 | 4-(4-phenoxyphenoxy)benzaldehyde | 96 | 110mg |
| 518 | methyl 6-methyl-1H-indole-2-carboxylate | 98 | 100mg |
| 519 | methyl 6-([1,1'-biphenyl]-3-yloxy)-1H-indole-2-carboxylate | 100 | 150mg |
| 520 | 4-(3-(3-hydroxypropyl)phenoxy)benzaldehyde | 94 | 150mg |
| 521 | 4-((2'-methyl-[1,1'-biphenyl]-4-yl)oxy)benzaldehyde | 100 | 150mg |
| 522 | 5-bromo-N-(3-nitrophenyl)pentanamide | 95 | 120mg |
| 523 | 1-(3-nitrophenyl)piperidin-2-one | 100 | 100mg |
| 524 | methyl 6-(4-phenoxyphenoxy)-1H-indole-2-carboxylate | 100 | 100mg |
| 525 | 3-(carboxymethyl)-7-methyl-1H-indole-2-carboxylic acid | 95 | 100mg |
| 526 | 1-(3-aminophenyl)piperidin-2-one | 95 | 200mg |
| 527 | 2-([1,1'-biphenyl]-4-yloxy)-4-fluorobenzaldehyde | 95 | 100mg |
| 528 | N-(5-bromo-2,3-dihydro-1H-inden-4-yl)pivalamide | 100 | 100 mg |
| 529 | 3-(6-chloro-5-((R)-3-methylmorpholino)pyridazin-3-yl)-8-oxa-3-azabicyclo[3.2.1]octane | 95 | 230 mg |
| 530 | 3-(6-chloro-5-(3,3-dimethylmorpholino)pyridazin-3-yl)-8-oxa-3-azabicyclo[3.2.1]octane | 96 | 220 mg |
| 531 | 5-(2-fluoropyridin-4-yl)-2,3-dihydro-1H-inden-4-amine | 85 | 372 mg |
| 532 | (R)-4-(7-iodopyrazolo[1,5-a]pyrimidin-5-yl)-3-methylmorpholine | 93 | 100 mg |
| 533 | 4-bromo-3,6-dichloropyridazine | 99 | 515 mg |
| 534 | 3,6-dichloro-4-(piperidin-1-yl)pyridazine | 98 | 204 mg |
| 535 | 3-ethyl 5-methyl 6-bromoimidazo[1,2-a]pyridine-3,5-dicarboxylate | 91 | 151 mg |
| 536 | (1R,5S)-3-(pyrazolo[1,5-a]pyrimidin-5-yl)-8-oxa-3-azabicyclo[3.2.1]octane | 96 | 136 mg |
| 537 | 3-ethyl 5-methyl 8-bromoimidazo[1,2-a]pyridine-3,5-dicarboxylate | 95 | 313 mg |
| 538 | N-(2,3-dihydro-1H-inden-4-yl)pivalamide | 100 | 100 mg |
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